网页Calicheamicin is a DNA synthesis inhibitor [1]. Calicheamicin is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups. PF-06647263 (anti-EFNA4-ADC) 是通过 hE22 赖氨酸残基与 AcButDMH-N-Ac-calicheamicin-γ1 连接子有效载荷 ...